Toxicity of cocaine versus methadone in brain development

(M.C. Nassogne and P.J. Courtoy, in collaboration with P. Gressens and Ph. Evrard, Hôpital Debré, Paris, France).

Using an in vitro system of mouse embryonic neuronal cell co-cultures, we have previously reported that the severe cerebral alterations found in children born to cocaine-addicted models could be due to inappropriate neuronal apoptosis (Nassogne et al., 1995, PNAS 92:11029-11033: Nassogne et al., 1997, J. Neurochem. 68:2442-2450; Ref. 19). The relevance of these observations in an animal model and the safety of methadone substitution in detoxification programs were assessed in pregnant mice. Methadone (40 mg/kg/day, i.e., 40-fold detoxification dosage) or cocaine (30 mg/kd/day, as in severe addiction) was injected into mice from day 8 to day 18 of gestation. Pre- and postnatal brain development was analyzed at the anatomical and microscopical levels, including by immunostaining of post-mitotic cells, neurites, and astrocytes. Prenatal mice exposure to cocaine caused neuronal misaddressing among neocortical layers, abnormal gliogenesis, and defective neuritic outgrowth and bundling. Methadone produced small-for-date offspring with normal brain development. In conclusion, supratherapeutic methadone doses induce intrauterine growth retardation in mice, but spare brain cytoarchitecture. In contrast, cocaine produces less growth retardation, but severely disturbs neocortical layering (Ref. 7).